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Discovery of 5-Nitro-6-thiocyanatopyrimidines as Inhibitors of Cryptococcus  neoformans and Cryptococcus gattii | ACS Medicinal Chemistry Letters
Discovery of 5-Nitro-6-thiocyanatopyrimidines as Inhibitors of Cryptococcus neoformans and Cryptococcus gattii | ACS Medicinal Chemistry Letters

Sortase A Inhibitors: Recent Advances and Future Perspectives | Journal of  Medicinal Chemistry
Sortase A Inhibitors: Recent Advances and Future Perspectives | Journal of Medicinal Chemistry

Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry  Letters
Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry Letters

Active Components of Essential Oils as Anti-Obesity Potential Drugs  Investigated by in Silico Techniques | Journal of Agricultural and Food  Chemistry
Active Components of Essential Oils as Anti-Obesity Potential Drugs Investigated by in Silico Techniques | Journal of Agricultural and Food Chemistry

ACS Medicinal Chemistry Letters | Vol 11, No 11
ACS Medicinal Chemistry Letters | Vol 11, No 11

a-Factor Analogues Containing Alkyne- and Azide-Functionalized Isoprenoids  Are Efficiently Enzymatically Processed and Retain Wild-Type Bioactivity |  Bioconjugate Chemistry
a-Factor Analogues Containing Alkyne- and Azide-Functionalized Isoprenoids Are Efficiently Enzymatically Processed and Retain Wild-Type Bioactivity | Bioconjugate Chemistry

Cytotoxic Effect of Silver Nanoparticles Synthesized by Green Methods in  Cancer | Journal of Medicinal Chemistry
Cytotoxic Effect of Silver Nanoparticles Synthesized by Green Methods in Cancer | Journal of Medicinal Chemistry

Automated De Novo Design in Medicinal Chemistry: Which Types of Chemistry  Does a Generative Neural Network Learn? | Journal of Medicinal Chemistry
Automated De Novo Design in Medicinal Chemistry: Which Types of Chemistry Does a Generative Neural Network Learn? | Journal of Medicinal Chemistry

Discovery of Potent and Selective 7-Azaindole Isoindolinone-Based PI3Kγ  Inhibitors | ACS Medicinal Chemistry Letters
Discovery of Potent and Selective 7-Azaindole Isoindolinone-Based PI3Kγ Inhibitors | ACS Medicinal Chemistry Letters

Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry  Letters
Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry Letters

Discovery and Preclinical Pharmacology of INE963, a Potent and Fast-Acting  Blood-Stage Antimalarial with a High Barrier to Resistance and Potential  for Single-Dose Cures in Uncomplicated Malaria | Journal of Medicinal  Chemistry
Discovery and Preclinical Pharmacology of INE963, a Potent and Fast-Acting Blood-Stage Antimalarial with a High Barrier to Resistance and Potential for Single-Dose Cures in Uncomplicated Malaria | Journal of Medicinal Chemistry

Discovery of a Novel Series of 7-Azaindole Scaffold Derivatives as PI3K  Inhibitors with Potent Activity | ACS Medicinal Chemistry Letters
Discovery of a Novel Series of 7-Azaindole Scaffold Derivatives as PI3K Inhibitors with Potent Activity | ACS Medicinal Chemistry Letters

Discovery of a 3-(4-Pyrimidinyl) Indazole (MLi-2), an Orally Available and  Selective Leucine-Rich Repeat Kinase 2 (LRRK2) Inhibitor that Reduces Brain  Kinase Activity | Journal of Medicinal Chemistry
Discovery of a 3-(4-Pyrimidinyl) Indazole (MLi-2), an Orally Available and Selective Leucine-Rich Repeat Kinase 2 (LRRK2) Inhibitor that Reduces Brain Kinase Activity | Journal of Medicinal Chemistry

Class 1 PI3K Clinical Candidates and Recent Inhibitor Design Strategies: A  Medicinal Chemistry Perspective | Journal of Medicinal Chemistry
Class 1 PI3K Clinical Candidates and Recent Inhibitor Design Strategies: A Medicinal Chemistry Perspective | Journal of Medicinal Chemistry

Discovery of Novel Cyanamide-Based Inhibitors of Cathepsin C | ACS  Medicinal Chemistry Letters
Discovery of Novel Cyanamide-Based Inhibitors of Cathepsin C | ACS Medicinal Chemistry Letters

Structure-Based Design of 3-(4-Aryl-1H-1,2,3-triazol-1-yl)-Biphenyl  Derivatives as P2Y14 Receptor Antagonists | Journal of Medicinal Chemistry
Structure-Based Design of 3-(4-Aryl-1H-1,2,3-triazol-1-yl)-Biphenyl Derivatives as P2Y14 Receptor Antagonists | Journal of Medicinal Chemistry

Applications of Deuterium in Medicinal Chemistry | Journal of Medicinal  Chemistry
Applications of Deuterium in Medicinal Chemistry | Journal of Medicinal Chemistry

Discovery of APD371: Identification of a Highly Potent and Selective CB2  Agonist for the Treatment of Chronic Pain | ACS Medicinal Chemistry Letters
Discovery of APD371: Identification of a Highly Potent and Selective CB2 Agonist for the Treatment of Chronic Pain | ACS Medicinal Chemistry Letters

LogD Contributions of Substituents Commonly Used in Medicinal Chemistry |  ACS Medicinal Chemistry Letters
LogD Contributions of Substituents Commonly Used in Medicinal Chemistry | ACS Medicinal Chemistry Letters

Discovery of Highly Selective Inhibitors of the Immunoproteasome Low  Molecular Mass Polypeptide 2 (LMP2) Subunit | ACS Medicinal Chemistry  Letters
Discovery of Highly Selective Inhibitors of the Immunoproteasome Low Molecular Mass Polypeptide 2 (LMP2) Subunit | ACS Medicinal Chemistry Letters

Journal of Medicinal Chemistry | Vol 65, No 2
Journal of Medicinal Chemistry | Vol 65, No 2

Synthesis of Thymoquinone–Artemisinin Hybrids: New Potent Antileukemia,  Antiviral, and Antimalarial Agents | ACS Medicinal Chemistry Letters
Synthesis of Thymoquinone–Artemisinin Hybrids: New Potent Antileukemia, Antiviral, and Antimalarial Agents | ACS Medicinal Chemistry Letters

Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry  Letters
Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry Letters

Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry  Letters
Metabolically Stable tert-Butyl Replacement | ACS Medicinal Chemistry Letters

Dominic Mata - QA/R&D Chemist - NHK Laboratories, Inc. | LinkedIn
Dominic Mata - QA/R&D Chemist - NHK Laboratories, Inc. | LinkedIn

Dehydrozingerone Inspired Styryl Hydrazine Thiazole Hybrids as Promising  Class of Antimycobacterial Agents | ACS Medicinal Chemistry Letters
Dehydrozingerone Inspired Styryl Hydrazine Thiazole Hybrids as Promising Class of Antimycobacterial Agents | ACS Medicinal Chemistry Letters

Publications - The Frantz Lab
Publications - The Frantz Lab